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Table 2 Antibiotics commonly used to treat biliary tract infections and their biliary penetration ability [46]

From: 2016 WSES guidelines on acute calculous cholecystitis

Good penetration efficiency (ABSCR > =1)

Low penetration efficiency (ABSCR <1)

Piperacillin/tazobactam (4.8)

Ceftriaxone (0.75)

Tigecycline (> 10)

Cefotaxime (0.23)

Amoxicillin/clavulanate (1.1)

Meropenem (0.38)

Ciprofloxacin (> 5)

Ceftazidime (0.18)

Ampicillin/Sulbactam (2.4)

Vancomycin (0.41)

Cefepime (2.04)

Amikacin (0.54)

Levofloxacin (1.6)

Gentamicin (0.30)

Penicillin “G” (>5)

 

Imipenem (1.01)

 
  1. ABSCR Antibiotics Bile/Serum Concentration Ratio